A simple efficient sequential one-pot intermolecular aza-Michael addition and intramolecular Buchwald-Hartwig α-arylation of amines: Synthesis of functionalized tetrahydroisoquinolines

Reddy, A G K and G, Satyanarayana (2012) A simple efficient sequential one-pot intermolecular aza-Michael addition and intramolecular Buchwald-Hartwig α-arylation of amines: Synthesis of functionalized tetrahydroisoquinolines. Tetrahedron, 68 (38). pp. 8003-8010. ISSN 0040-4020

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Abstract

An efficient one-pot sequential intermolecular aza-Michael addition and Pd-catalyzed intramolecular Buchwald-Hartwig α-arylation of secondary amines have been investigated, for the synthesis of tetrahydroisoquinolines. This method is simple and furnished products in very good yield and also successfully applied for the synthesis of novel aza-spirotricylcic ethers

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IITH Creators:

IITH Creators	ORCiD
G, Satyanarayana	UNSPECIFIED

Item Type:

Article

Additional Information:

This research work is dedicated to Professor Dr. Günter Helmchen, Organisch-Chemisches Institut der Universität Heidelberg. We thank Dr. P.C. Ravi Kumar and Dr. Santosh J. Gharpure for valuable suggestions. A.G.K. thanks CSIR, New Delhi, for the award of research fellowship.

Uncontrolled Keywords:

α-Arylation; Aza-Michael; Pd-catalysis; Sequential one-pot; Tetrahydroisoquinolines

Subjects:

?? sub5.8 ??

Divisions:

Department of Chemistry

Depositing User:

Team Library

Date Deposited:

11 Nov 2014 04:09

Last Modified:

24 Sep 2015 10:28